SCHEMBL29138513

SCHEMBL29138513

COC(=O)C(=O)c1c[nH]c2cccc(OCc3ccccc3)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.52
EDNRA P25101 1/20 0.46
SRD5A2 P31213 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.43
BRD4 O60885 1/20 0.43
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
GABRA4 P48169 1/20 0.42
GABRE P78334 1/20 0.42
GABRA6 Q16445 1/20 0.42
GABRG1 Q8N1C3 1/20 0.42
GABRG3 Q99928 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23805228 0.87 HTR2A (0.51) HTR2AEDNRASRD5A2BRD4GABRP
SCHEMBL30960130 0.86 HTR2A (0.52) HTR2AEDNRASRD5A2SGMS2PTGER1
SCHEMBL11067101 0.85 HTR2A (0.53) HTR2AEDNRASRD5A2SGMS2ALDH1A1
SCHEMBL7390324 0.85 HTR2A (0.55) HTR2AEDNRASRD5A2SGMS2PTGER1
SCHEMBL12558840 0.85 HTR2A (0.57) HTR2AEDNRASRD5A2ABCG2BRD4
SCHEMBL1163120 0.84 PTGER1 (0.41) SRD5A2PTGER1ALDH1A1HPGDMDH2
SCHEMBL31027232 0.84 HTR2A (0.48) HTR2ASRD5A2ABCG2GABRPGABRD
SCHEMBL31614675 0.83 NPC1 (0.50) HTR2AGABRPGABRDGABRA1GABRB1
SCHEMBL23805270 0.83 HTR2A (0.52) HTR2AEDNRASRD5A2GABRPGABRD
SCHEMBL6031099 0.82 MTNR1A (0.52) HTR2AGABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119698412-A 5-HT2A receptor agonist, and preparation method and application thereof 上海翊石医药科技有限公司 2025-03-25 CN disclosed
WO-2025021120-A1 5-HT2A RECEPTOR AGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊石医药科技有限公司 2025-01-30 WO disclosed
CN-117069720-A 5-HT 2A Receptor agonist, preparation method and application thereof 上海翊石医药科技有限公司 2023-11-17 CN disclosed