SCHEMBL291388

SCHEMBL291388

COCCOc1ccccc1N1CC(C)(C)N(C(=O)OC(C)(C)C)CC1=O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
REN P00797 10/20 0.48
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
KDM1A O60341 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
P2RX3 P56373 1/20 0.33
DRD2 P14416 1/20 0.33
GAA P10253 1/20 0.33
HTR6 P50406 1/20 0.33
BCHE P06276 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL291856 0.95 REN (0.49) RENHDAC1HDAC6DDB1CRBN
SCHEMBL293123 0.91 REN (0.48) RENHDAC1HDAC6DDB1CRBN
SCHEMBL293228 0.87 REN (0.44) RENALDH1A1DRD2BCHE
SCHEMBL291213 0.86 SNRNP200 (0.41) RENHDAC1HDAC6GAAHTR6
SCHEMBL292245 0.81 NR1H2 (0.39) RENHDAC1HDAC6KDM1AGAA
SCHEMBL292987 0.81 MAPT (0.41) RENHDAC1HDAC6DDB1CRBN
SCHEMBL291695 0.80 REN (0.45) REN
SCHEMBL27776020 0.79 HDAC1 (0.36) RENHDAC1HDAC6KDM1ABCHE
SCHEMBL292539 0.77 NR1H2 (0.45) RENALDH1A1GAABCHE
SCHEMBL292325 0.77 DRD2 (0.42) RENKDM4EALDH1A1TDP1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101511799-B Cyclic amine compound DAIICHI SANKYO CO LTD 2012-05-30 CN disclosed
US-8158790-B2 Cyclic amine compound DAIICHI SANKYO COMPANY, LIMITED (JP) 2012-04-17 US disclosed
EP-2036896-B1 CYCLIC AMINE COMPOUND DAIICHI SANKYO CO LTD (JP) 2012-03-14 EP disclosed
US-20090286807-A1 CYCLIC AMINE COMPOUND DAIICHI SANKYO COMPANY, LIMITED (JP) 2009-11-19 US disclosed
CN-101511799-A Cyclic amine compound DAIICHI SANKYO CO LTD (JP) 2009-08-19 CN disclosed
EP-2036896-A1 CYCLIC AMINE COMPOUND Daiichi Sankyo Company, Limited (JP) 2009-03-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090286807-A1 CYCLIC AMINE COMPOUND HRH3, HRH4, H1-0 REN 35/4885HDAC1 792/4885HDAC6 3636/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.