SCHEMBL29139855

SCHEMBL29139855

O=C(O)c1ccnc(N2CC(O)C2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.61
PROKR1 Q8TCW9 1/20 0.54
KDM4C Q9H3R0 17/20 0.50
KDM5A P29375 14/20 0.50
KDM5B Q9UGL1 13/20 0.50
KDM4A O75164 4/20 0.49
KDM2B Q8NHM5 5/20 0.49
KDM4E B2RXH2 1/20 0.47
KDM6B O15054 1/20 0.47
TET3 O43151 1/20 0.47
BBOX1 O75936 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
KDM5C P41229 1/20 0.47
ASPH Q12797 1/20 0.47
KDM4D Q6B0I6 1/20 0.47
TET2 Q6N021 1/20 0.47
ALKBH5 Q6P6C2 1/20 0.47
KDM7A Q6ZMT4 1/20 0.47
KDM8 Q8N371 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30775157 1.00 PIK3CA (0.61) PIK3CAPROKR1KDM4CKDM5AKDM5B
Nitrous Acid SCHEMBL29139860 0.94 PIK3CA (0.56) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL3743262 0.84 PIK3CA (0.67) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL19202594 0.82 PROKR1 (0.53) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL30378524 0.82 PROKR1 (0.53) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL31143236 0.80 PIK3CA (0.74) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL1516867 0.80 PIK3CA (0.74) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL29139858 0.80 PROKR1 (0.48) PIK3CAPROKR1KDM4CKDM5AKDM5B
Hydrochloric Acid SCHEMBL1252523 0.79 PIK3CA (0.72) PIK3CAPROKR1KDM4CKDM5AKDM5B
SCHEMBL1255519 0.79 PIK3CA (0.72) PIK3CAPROKR1KDM4CKDM5AKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924266-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-117924267-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-109476636-B Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-01-09 CN disclosed