SCHEMBL29139857

SCHEMBL29139857

O=NOC(=O)c1ccnc(N2CC(=O)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.44
HRH3 Q9Y5N1 2/20 0.36
MAPK13 O15264 1/20 0.36
KDM4C Q9H3R0 6/20 0.35
KDM2B Q8NHM5 3/20 0.35
USP30 Q70CQ3 1/20 0.34
KDM5A P29375 4/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KDM5B Q9UGL1 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
KDM4A O75164 1/20 0.34
PROKR1 Q8TCW9 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALOX15 P16050 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14641897 0.83 KDM4C (0.50) PIK3CAHRH3KDM4CKDM5ANPC1
SCHEMBL29139858 0.82 PROKR1 (0.48) PIK3CAHRH3MAPK13KDM4CUSP30
Nitrous Acid SCHEMBL29139859 0.80 PIK3CA (0.57) PIK3CAKDM4CKDM2BKDM5AKDM5B
SCHEMBL29139863 0.79 PIK3CA (0.63) PIK3CAKDM4CKDM2BKDM5AKDM5B
SCHEMBL30775160 0.79 PIK3CA (0.63) PIK3CAKDM4CKDM2BKDM5AKDM5B
SCHEMBL28781584 0.72 NPC1 (0.42) KDM4CKDM5ANPC1RAB9AKDM5B
SCHEMBL28404952 0.71 MAPT (0.44) KDM4CNPC1RAB9AALDH1A1POLB
SCHEMBL29072870 0.71 KMT2A (0.43) KDM4CNPC1RAB9AALDH1A1POLB
SCHEMBL28381981 0.71 NPC1 (0.39) KDM4CKDM5ANPC1RAB9AKDM5B
SCHEMBL28394531 0.71 GABRP (0.58) KDM4CNPC1RAB9AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924266-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-117924267-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-109476636-B Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-01-09 CN disclosed