SCHEMBL29139869

SCHEMBL29139869

Cc1nc(N2CC(O)(c3ccc(O[Si](C)(C)C(C)(C)C)cc3Cl)C2)c(F)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 19/20 0.45
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
HSD17B13 Q7Z5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19699379 0.81 NR1H4 (0.48) NR1H4
SCHEMBL19689515 0.78 NR1H4 (0.51) NR1H4
SCHEMBL30775168 0.78 NR1H4 (0.51) NR1H4
SCHEMBL22320341 0.77 CA12 (0.39) NR1H4CA12CA1CA9HSD17B13
SCHEMBL19690343 0.76 NR1H4 (0.44) NR1H4
SCHEMBL29216000 0.75 NR1H4 (0.54) NR1H4HSD17B13
SCHEMBL30775154 0.75 NR1H4 (0.54) NR1H4HSD17B13
SCHEMBL29139862 0.73 NR1H4 (0.77) NR1H4HSD17B13
SCHEMBL29736070 0.72 MET (0.37) CA12CA1CA9
SCHEMBL19689482 0.72 MET (0.37) CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117924266-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-117924267-A Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-04-26 CN disclosed
CN-109476636-B Compounds that modulate FXR (NR 1H 4) 吉利德科学公司 2024-01-09 CN disclosed