SCHEMBL2914083

SCHEMBL2914083

CC(C)(C)OC(=O)c1cn(CCCNc2ccc([N+](=O)[O-])c(N)n2)cc1-c1ccc(F)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 2/20 0.35
GSK3B P49841 5/20 0.35
GSK3A P49840 4/20 0.35
QPCT Q16769 3/20 0.33
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.32
CDK1 P06493 2/20 0.32
KCNQ3 O43525 1/20 0.31
KCNQ2 O43526 1/20 0.31
ABCB11 O95342 1/20 0.31
ESR1 P03372 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31
NFKB1 P19838 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904943 0.93 GSK3B (0.35) GSK3BGSK3ALMNACDK1CCNB2
SCHEMBL2905411 0.92 GSK3B (0.35) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL2910908 0.92 GSK3B (0.41) GSK3BGSK3AHTTLMNACDK1
SCHEMBL2904037 0.91 GSK3B (0.34) METGSK3BGSK3ACDK1AXL
SCHEMBL2910444 0.91 MAPT (0.35) GSK3BGSK3AHTTLMNACYP1A2
SCHEMBL2912809 0.90 GSK3B (0.37) METGSK3BGSK3ACDK1CCNB2
SCHEMBL2912022 0.90 GSK3B (0.34) GSK3BGSK3ACDK1AXLMERTK
SCHEMBL2910224 0.88 GSK3B (0.42) GSK3BGSK3AHTTLMNACDK1
SCHEMBL2911792 0.88 GSK3B (0.36) METGSK3BGSK3AQPCTHTT
SCHEMBL2912012 0.86 GSK3A (0.41) GSK3BGSK3AHTTCDK1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed