SCHEMBL29151978

SCHEMBL29151978

Cc1ncnc2c(OCc3ccc(C(=O)OC(C)(C)C)cc3)cc(Br)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.41
HDAC1 Q13547 5/20 0.41
CCR5 P51681 1/20 0.40
SMPD1 P17405 1/20 0.37
MAPT P10636 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 1/20 0.37
PTGER1 P34995 1/20 0.36
MAOB P27338 2/20 0.35
RXRA P19793 3/20 0.35
RXRB P28702 3/20 0.35
RXRG P48443 3/20 0.35
MAOA P21397 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30631225 0.85 RXRA (0.49) PIK3CAHDAC1RAB9ARXRARXRB
SCHEMBL29151981 0.85 RXRA (0.49) PIK3CAHDAC1RAB9ARXRARXRB
SCHEMBL29152006 0.85 MEN1 (0.36) PIK3CAHDAC1L3MBTL1MEN1KMT2A
SCHEMBL29152026 0.77 HDAC1 (0.57) PIK3CAHDAC1MAPTLMNARAB9A
SCHEMBL29152021 0.76 PIK3CA (0.45) PIK3CAHDAC1
SCHEMBL28457959 0.74 CA12 (0.41) PIK3CAHDAC1ATM
SCHEMBL30631181 0.73 ELANE (0.41) PIK3CAHDAC1MAPTLMNARAB9A
SCHEMBL28460294 0.73 CA12 (0.42) PIK3CAHDAC1CYP2C19ATM
SCHEMBL28457788 0.73 PIK3CA (0.40) PIK3CAHDAC1
SCHEMBL28445733 0.72 CA12 (0.43) PIK3CAHDAC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116987061-A 4-methyl quinazoline derivative, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2023-11-03 CN disclosed