SCHEMBL29151981

SCHEMBL29151981

Cc1ncnc2c(OCc3ccc(C(=O)O)cc3)cc(Br)cc12

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXRA P19793 9/20 0.49
RXRB P28702 8/20 0.49
RXRG P48443 5/20 0.49
FOLH1 Q04609 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.44
PIK3CA P42336 2/20 0.44
HDAC1 Q13547 2/20 0.44
PPARA Q07869 1/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.42
SLC26A4 O43511 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
MAP4K4 O95819 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30631225 1.00 RXRA (0.49) RXRARXRBRXRGFOLH1MRGPRX4
SCHEMBL29151978 0.85 PIK3CA (0.41) RXRARXRBRXRGPIK3CAHDAC1
SCHEMBL29152026 0.83 HDAC1 (0.57) PIK3CAHDAC1HPGDNPC1RAB9A
SCHEMBL29152046 0.83 RXRA (0.44) RXRARXRBRXRGPIK3CAHDAC1
SCHEMBL30631223 0.83 RXRA (0.44) RXRARXRBRXRGPIK3CAHDAC1
SCHEMBL30631181 0.75 ELANE (0.41) PIK3CAHDAC1HPGDNPC1RAB9A
SCHEMBL29152063 0.75 PIK3CA (0.49) PIK3CAHDAC1
SCHEMBL30631159 0.75 PIK3CA (0.49) PIK3CAHDAC1
SCHEMBL28460296 0.73 ALDH1A1 (0.48) PIK3CAHDAC1HPGDSMN1; SMN2MEN1
SCHEMBL19249082 0.71 RXRA (0.48) RXRARXRBRXRGFOLH1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116987061-A 4-methyl quinazoline derivative, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2023-11-03 CN disclosed