SCHEMBL29169136

SCHEMBL29169136

O=C1CNCCN1c1ncc(C(F)(F)F)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.36
PARP1 P09874 1/20 0.34
SCN9A Q15858 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
APAF1 O14727 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PIM1 P11309 1/20 0.33
LCAT P04180 1/20 0.33
SCN7A Q01118 1/20 0.33
KCNH2 Q12809 2/20 0.33
TIPARP Q7Z3E1 1/20 0.33
ADRB2 P07550 1/20 0.32
NCF1 P14598 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1578382 0.81 MAPT (0.48) ADRB1SMN1; SMN2ALDH1A1KDM4EAPAF1
Hydrochloric Acid SCHEMBL1962520 0.80 MAPT (0.47) ADRB1SMN1; SMN2ALDH1A1KDM4EAPAF1
SCHEMBL6767507 0.77 ALDH1A1 (0.48) SMN1; SMN2ALDH1A1KDM4EMAPTPIM1
SCHEMBL9199798 0.76 SLC6A2 (0.36) PARP1ALDH1A1KDM4EPIM1SLC6A2
SCHEMBL3068463 0.75 ADRB1 (0.42) ADRB1SCN9AALDH1A1MAPTLCAT
SCHEMBL8195822 0.75 SLC6A2 (0.46) ADRB1SCN9AALDH1A1MAPTSLC6A2
SCHEMBL28817805 0.75 ADRB1 (0.56) ADRB1SCN9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL3081103 0.74 ADRB1 (0.62) ADRB1ALDH1A1MAPTPIM1ADRB2
SCHEMBL3922344 0.74 ALDH1A1 (0.53) ADRB1PARP1SMN1; SMN2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL21522534 0.72 ALDH1A1 (0.56) ADRB1SMN1; SMN2ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117377665-A PARP7 inhibitor and application thereof 北京华森英诺生物科技有限公司 2024-01-09 CN disclosed