SCHEMBL2917019

SCHEMBL2917019

CCC(SC(c1ccc(C#N)cc1)c1c[nH]cn1)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.35
ALOX5 P09917 4/20 0.35
PPARG P37231 2/20 0.35
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
CYP19A1 P11511 2/20 0.32
HSD11B1 P28845 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
EGLN1 Q9GZT9 2/20 0.31
PKM P14618 1/20 0.31
PPARA Q07869 1/20 0.31
S1PR1 P21453 2/20 0.30
S1PR3 Q99500 2/20 0.30
HTT P42858 2/20 0.30
SLC1A3 P43003 1/20 0.30
SLC1A2 P43004 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910903 0.80 HTT (0.42) GAAKDM4EMAPTL3MBTL1CYP19A1
SCHEMBL2910386 0.70 TOP2A (0.37) CYP19A1
SCHEMBL12130734 0.66 PGR (0.39) MAPTALDH1A1CYP19A1HRH3
SCHEMBL5891827 0.65 CYP19A1 (0.36) CYP19A1
SCHEMBL9090439 0.65 CYP19A1 (0.55) CYP19A1
SCHEMBL31554349 0.65 AKR1C3 (0.33)
SCHEMBL2474521 0.65 GAA (0.48) GAAKDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL9090407 0.64 CYP19A1 (0.62) CYP19A1SLC1A3SLC1A2
SCHEMBL7281806 0.63 SMN1; SMN2 (0.31)
Hydrochloric Acid SCHEMBL6781604 0.61 PTGS2 (0.53) ALOX5GAAKDM4EMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004657-B1 CONDENSED IMIDAZOLE DERIVATIVES AS ALDOSTERONE SYNTHASE INHIBITORS NOVARTIS AG (CH) 2010-09-01 EP disclosed