SCHEMBL29174281

SCHEMBL29174281

CC(=O)Oc1ccc(C(C)(C)C)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.50
MAPT P10636 3/20 0.50
POLB P06746 1/20 0.50
PKM P14618 1/20 0.50
ALDH1A1 P00352 3/20 0.46
GLA P06280 2/20 0.46
F2 P00734 1/20 0.46
HPGD P15428 1/20 0.46
CYP3A4 P08684 3/20 0.41
ELANE P08246 3/20 0.41
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 3/20 0.39
ABCB11 O95342 1/20 0.39
ESR1 P03372 1/20 0.39
ADRA2A P08913 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
PDE4A P27815 1/20 0.39
ADRA1A P35348 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27526965 0.84 POLB (0.49) LMNAMAPTPOLBPKMALDH1A1
SCHEMBL29177428 0.84 KMT2A (0.40) MAPTPOLBPKMALDH1A1GLA
SCHEMBL29163724 0.79 MAPT (0.60) LMNAMAPTPKMALDH1A1HSD17B10
SCHEMBL14062418 0.78 MAPT (0.59) LMNAMAPTALDH1A1HSD17B10KMT2A
SCHEMBL29123252 0.77 SMN1; SMN2 (0.57) LMNAMAPTPOLBALDH1A1CYP2C9
SCHEMBL3787327 0.76 SMN1; SMN2 (0.60) LMNAMAPTALDH1A1TSHRKMT2A
SCHEMBL11790413 0.76 KMT2A (0.57) LMNAMAPTPOLBPKMALDH1A1
SCHEMBL28452003 0.76 SMN1; SMN2 (0.63) LMNAMAPTPOLBALDH1A1HSD17B10
SCHEMBL27337562 0.76 ALDH1A1 (0.50) LMNAMAPTPOLBPKMALDH1A1
SCHEMBL10220768 0.75 CA12 (0.42) LMNAMAPTPOLBPKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396474-A Plasma kallikrein inhibitors 武田药品工业株式会社 2024-01-12 CN disclosed
CN-116507332-A Octahydroisoquinolinyl derivatives UCB生物制药有限责任公司 2023-07-28 CN disclosed