SCHEMBL29178351

SCHEMBL29178351

CNC(=O)C(CCCc1ccc(O)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.54
CTSS P25774 5/20 0.54
MMP1 P03956 3/20 0.53
MMP3 P08254 3/20 0.53
MMP9 P14780 2/20 0.53
PPARA Q07869 3/20 0.46
CA2 P00918 2/20 0.46
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
CA1 P00915 1/20 0.45
SIRT5 Q9NXA8 1/20 0.44
PPARG P37231 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25139698 1.00 CTSK (0.54) CTSKCTSSMMP1MMP3MMP9
SCHEMBL24814567 0.89 MMP3 (0.64) CTSKCTSSMMP1MMP3MMP9
SCHEMBL29178423 0.89 MMP3 (0.64) CTSKCTSSMMP1MMP3MMP9
SCHEMBL31407745 0.88 CTSK (0.56) CTSKCTSSPPARAPPARG
SCHEMBL29055935 0.88 CTSK (0.56) CTSKCTSSPPARAPPARG
SCHEMBL29178415 0.87 PPARA (0.52) CTSKCTSSMMP1MMP3MMP9
SCHEMBL24814570 0.87 PPARA (0.52) CTSKCTSSMMP1MMP3MMP9
SCHEMBL24812414 0.87 MMP3 (0.52) CTSKCTSSMMP1MMP3MMP9
SCHEMBL29178360 0.87 MMP3 (0.52) CTSKCTSSMMP1MMP3MMP9
SCHEMBL25312195 0.86 CTSK (0.52) CTSKCTSSPPARACA2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117561058-A CDK2 inhibitors and methods of use thereof 塞迪拉治疗股份有限公司 2024-02-13 CN disclosed