SCHEMBL2918183

SCHEMBL2918183

COCCn1c(-c2cc(OC)c(OC)c(OC)c2Br)nc2sc3c(O)cccc3c2c1=O

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.78
SMN1; SMN2 Q16637 4/20 0.44
LMNA P02545 1/20 0.44
ALDH1A1 P00352 7/20 0.41
RXFP1 Q9HBX9 2/20 0.40
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
ABCC1 P33527 1/20 0.37
MAPT P10636 3/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
STAT3 P40763 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
MAPK10 P53779 1/20 0.36
CTSV O60911 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2915813 0.89 HSD11B1 (0.79) HSD11B1SMN1; SMN2LMNAALDH1A1RXFP1
SCHEMBL2926603 0.87 HSD11B1 (1.00) HSD11B1SMN1; SMN2ALDH1A1RXFP1HSD17B10
SCHEMBL2924044 0.83 HSD11B1 (0.69) HSD11B1SMN1; SMN2LMNAALDH1A1HSD17B10
SCHEMBL1820439 0.81 HSD11B1 (0.62) HSD11B1SMN1; SMN2LMNAALDH1A1MEN1
SCHEMBL2922695 0.80 HSD11B1 (0.87) HSD11B1ALDH1A1RXFP1HSD17B10MEN1
SCHEMBL1821489 0.79 HSD11B1 (0.85) HSD11B1SMN1; SMN2LMNAALDH1A1RXFP1
SCHEMBL2915776 0.79 HSD11B1 (0.84) HSD11B1SMN1; SMN2ALDH1A1HSD17B10MEN1
SCHEMBL2924374 0.78 HSD11B1 (0.63) HSD11B1SMN1; SMN2LMNAALDH1A1RXFP1
SCHEMBL1819589 0.77 HSD11B1 (0.58) HSD11B1SMN1; SMN2LMNAALDH1A1MEN1
SCHEMBL2922023 0.77 HSD11B1 (0.57) HSD11B1SMN1; SMN2LMNAALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1635839-B1 BENZO[4,5]THIENO[2,3-D]PYRIMIDIN-4-ONES AND THEIR USE IN THERAPY ABBOTT HEALTHCARE PRODUCTS BV (NL) 2010-09-01 EP disclosed
US-7524853-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2009-04-28 US disclosed
US-7524853-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2009-04-28 US disclosed
US-7524853-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2009-04-28 US disclosed
US-7465739-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2008-12-16 US disclosed
US-7465739-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2008-12-16 US disclosed
US-7465739-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2008-12-16 US disclosed
EP-1635839-A2 BENZO[4,5]THIENO[2,3-D]PYRIMIDIN-4-ONES AND THEIR USE IN THERAPY Solvay Pharmaceuticals B.V. (NL) 2006-03-22 EP disclosed
US-20050176742-A1 Novel compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2005-08-11 US disclosed
WO-2005032527-A2 BENZO (4, 5) THIENO (2, 3-D) PYRIMIDIN-4-ONES AND THEIR USE IN THERAPY SOLVAY PHARMACEUTICALS B.V. (NL) 2005-04-14 WO disclosed
US-20050038053-A1 Novel compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2005-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176742-A1 Novel compounds and their use in therapy HSD17B11, HSD17B2, HSD17B1 HSD11B1 10/4885SMN1; SMN2 3338/4885LMNA 4510/4885
US-20050038053-A1 Novel compounds and their use in therapy HSD17B11, HSD17B2, HSD17B1 HSD11B1 10/4885SMN1; SMN2 3338/4885LMNA 4510/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.