Pinocembrin

Pinocembrin

SCHEMBL291899

O=C1CC(c2ccccc2)Oc2cc(O)cc(O)c21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 1.00
CYP3A4 P08684 5/20 1.00
CYP1A1 P04798 4/20 1.00
CYP1A2 P05177 4/20 1.00
CYP1B1 Q16678 4/20 1.00
CYP2C19 P33261 3/20 1.00
HSD17B10 Q99714 3/20 1.00
MAPT P10636 3/20 1.00
MEN1 O00255 2/20 1.00
CYP2C9 P11712 2/20 1.00
KMT2A Q03164 2/20 1.00
CYP2D6 P10635 1/20 1.00
TTR P02766 4/20 0.82
PSMB5 P28074 3/20 0.82
CA12 O43570 2/20 0.82
SLCO2B1 O94956 2/20 0.82
CA4 P22748 2/20 0.82
CA7 P43166 2/20 0.82
ALOX12 P18054 1/20 0.82
ESR1 P03372 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pinocembrin SCHEMBL30186539 1.00 CYP19A1 (1.00) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
(R)-Pinocembrin SCHEMBL10080882 1.00 CYP19A1 (1.00) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Pinocembrin SCHEMBL10026578 1.00 CYP19A1 (1.00) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Pinocembrin SCHEMBL2484359 0.99 CYP19A1 (0.97) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Pinocembrin SCHEMBL2232882 0.97 CYP19A1 (0.95) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Pinocembrin SCHEMBL3437711 0.94 CYP19A1 (0.88) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Naringenin SCHEMBL1333765 0.90 CYP19A1 (0.81) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Pinocembrin SCHEMBL17651823 0.90 CYP19A1 (0.81) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Naringenin SCHEMBL72954 0.90 CYP19A1 (0.81) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1
Naringenin SCHEMBL1048136 0.90 CYP19A1 (1.00) CYP19A1CYP3A4CYP1A1CYP1A2CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3061 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402197-B Vitex negundo extract and preparation method thereof and identification method of Vitex negundo honey 江苏蜂奥生物科技有限公司 2026-05-15 CN claimed
CN-122005744-A Quality marker for preventing and treating kidney-yang deficiency by using medicinal and edible formula composition, and preparation method and application thereof 广西壮族自治区中医药研究院 2026-05-12 CN claimed
WO-2026088186-A1 FERMENTED AND DEHYDRATED ALOE GEL PRODUCT AND PROCESS FOR THE PREPARATION THEREOF YOSHAY IDO MOSHE (IL) 2026-04-30 WO claimed
US-20260102359-A1 COMBINATION TREATMENT OF DERMAL AND TRANSDERMAL FIBROTIC DISEASES, DISORDERS AND ASSOCIATED PAIN AND INFLAMMATION ERESINA LLC (US) 2026-04-16 US claimed
US-20260091016-A1 Composition for preventing and/or combating neuroinflammation, particularly in neuropsychiatric and neurological diseases BEE TERAPI (FR) 2026-04-02 US claimed
EP-3346842-B1 STABLE INOCULANT COMPOSITIONS AND METHODS FOR PRODUCING SAME NOVONESIS PLANT BIOSOLUTIONS AS (DK) 2026-03-25 EP claimed
CN-121570478-A Antibacterial composition with synergistic effect of pinocembrin and aminoglycoside drugs and application thereof 中国农业大学三亚研究院 2026-02-27 CN claimed
EP-4062903-B1 METHOD FOR PRODUCING AN ACTIVE COMPLEX FROM LYMANTRIA DISPAR LARVAE CIUHRII CESLAV (MD) 2026-02-18 EP claimed
US-12532902-B2 Compositions and methods for taste modulation GIVAUDAN SA (CH) 2026-01-27 US claimed
EP-4656062-A1 SALTY TASTE/UMAMI ENHANCER AJINOMOTO CO., INC. (JP) 2025-12-03 EP claimed
US-5591771-A Use of propolis components as an adjuvant Fockerman, Michel (SE) 1997-01-07 US claimed
EP-0719554-A1 Chondroprotective flavonoids Kureha Chemical Industry Co., Ltd. (JP) 1996-07-03 EP claimed
EP-0707851-A2 Benzopyran phenol derivates for use as antibacterial, antiviral or immunostimulating agents Fockerman, Jasmine (SE) 1996-04-24 EP claimed
US-5449794-A Benzopyran phenol derivatives for use as antibacterial agents Fockerman, Jasmine (SE) 1995-09-12 US claimed
EP-0633022-A2 Chondroprotective flavones KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-01-11 EP claimed
EP-0571491-A1 BENZOPYRAN PHENOL DERIVATES FOR USE AS ANTIBACTERIAL, ANTIVIRAL OR IMMUNOSTIMULATING AGENTS. FOCKERMAN JASMINE (SE) 1993-12-01 EP claimed
WO-1992014458-A1 BENZOPYRAN PHENOL DERIVATES FOR USE AS ANTIBACTERIAL, ANTIVIRAL OR IMMUNOSTIMULATING AGENTS FOCKERMAN, JASMINE (SE) 1992-09-03 WO claimed
EP-0499015-A1 Benzopyran phenol derivates for use as antibacterial, antiviral or immunostimulating agents Fockerman, Jasmine (SE) 1992-08-19 EP claimed
US-4617293-A Flavonoid phosphate salts of aminoglycoside antibiotics MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1986-10-14 US claimed
US-4105675-A REDUCING ACYLATED FLAVANONE WITH ALKALI BOROHYDRIDE TO REMOVE OXYGEN FUNCTION AT 4-POSITION; OXIDIZING WITH HALOGENATED BENZOQUINONE TO FORM SALT THE COCA-COLA COMPANY (US) 1978-08-08 US claimed