SCHEMBL29190702

SCHEMBL29190702

CN1CCN(c2n[nH]c3cc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5NS(C)(=O)=O)n4)ccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 6/20 0.53
FLT3 P36888 2/20 0.53
EGFR P00533 6/20 0.52
BRD4 O60885 4/20 0.49
PTK2 Q05397 2/20 0.46
ULK1 O75385 1/20 0.46
ROS1 P08922 1/20 0.45
CDK1 P06493 1/20 0.44
CDK4 P11802 1/20 0.44
CDK2 P24941 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190646 0.91 ALK (0.47) ALKFLT3EGFRBRD4PTK2
SCHEMBL29190605 0.89 ALK (0.67) ALKFLT3EGFRBRD4ROS1
SCHEMBL30833773 0.87 BRD4 (0.47) ALKFLT3EGFRBRD4PTK2
SCHEMBL29190535 0.87 ALK (0.53) ALKFLT3EGFRBRD4PTK2
SCHEMBL29190604 0.86 ALK (0.52) ALKFLT3EGFRBRD4ROS1
SCHEMBL30833633 0.85 EGFR (0.47) ALKFLT3EGFRBRD4PTK2
SCHEMBL29190602 0.85 ALK (0.53) ALKFLT3EGFRBRD4ROS1
SCHEMBL29190617 0.80 ALK (0.68) ALKFLT3EGFRPTK2ULK1
SCHEMBL29190594 0.80 PTK2 (0.52) ALKEGFRPTK2ULK1CDK1
SCHEMBL29190521 0.75 PTK2 (0.56) ALKFLT3EGFRPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed