SCHEMBL30833633

SCHEMBL30833633

CN1CCN(c2n[nH]c3cc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5CN[SH](=O)=O)n4)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.47
ULK1 O75385 2/20 0.44
BRD4 O60885 2/20 0.43
PTK2 Q05397 9/20 0.42
ALK Q9UM73 2/20 0.42
WEE1 P30291 1/20 0.42
CDK1 P06493 1/20 0.42
CDK4 P11802 1/20 0.42
CDK2 P24941 1/20 0.42
PTK2B Q14289 4/20 0.42
KDR P35968 1/20 0.41
AURKB Q96GD4 1/20 0.41
FLT3 P36888 3/20 0.41
BTK Q06187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833801 0.91 EGFR (0.42) EGFRULK1BRD4PTK2ALK
SCHEMBL30833773 0.87 BRD4 (0.47) EGFRULK1BRD4PTK2ALK
SCHEMBL29190716 0.87 FGFR1 (0.44) EGFRULK1PTK2ALKWEE1
SCHEMBL29190702 0.85 ALK (0.53) EGFRULK1BRD4PTK2ALK
SCHEMBL29190553 0.84 INSR (0.46) EGFRALKKDRFLT3BTK
SCHEMBL30833808 0.81 PTK2 (0.47) ULK1PTK2CDK1CDK4CDK2
SCHEMBL30833699 0.81 EGFR (0.49) EGFRULK1PTK2ALKCDK2
SCHEMBL30833721 0.79 BRD4 (0.42) EGFRULK1BRD4PTK2ALK
SCHEMBL30833740 0.78 PTK2 (0.50) ULK1PTK2CDK1CDK4CDK2
SCHEMBL29190646 0.77 ALK (0.47) EGFRULK1BRD4PTK2ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed