SCHEMBL29190604

SCHEMBL29190604

CC(c1cnc(Nc2ccc3c(N4CCN(C)CC4)n[nH]c3c2)nc1Nc1ccccc1NS(C)(=O)=O)[Si](C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 9/20 0.52
FLT3 P36888 2/20 0.52
ROS1 P08922 2/20 0.47
EGFR P00533 6/20 0.46
BRD4 O60885 2/20 0.44
GLO1 Q04760 1/20 0.41
MAP3K7 O43318 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190605 0.88 ALK (0.67) ALKFLT3ROS1EGFRBRD4
SCHEMBL29190535 0.86 ALK (0.53) ALKFLT3ROS1EGFRBRD4
SCHEMBL29190702 0.86 ALK (0.53) ALKFLT3ROS1EGFRBRD4
SCHEMBL29190602 0.85 ALK (0.53) ALKFLT3ROS1EGFRBRD4
SCHEMBL29190617 0.81 ALK (0.68) ALKFLT3EGFR
SCHEMBL29190646 0.77 ALK (0.47) ALKFLT3ROS1EGFRBRD4
SCHEMBL29190656 0.75 BRD4 (0.57) ALKFLT3ROS1EGFRBRD4
SCHEMBL29190626 0.74 EGFR (0.52) ALKFLT3EGFR
SCHEMBL29190585 0.74 CDK9 (0.54) ALKFLT3EGFRMAP3K7MAPK1
SCHEMBL29190551 0.73 ALK (0.67) ALKFLT3EGFRGLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed