SCHEMBL291979

SCHEMBL291979

C=Cc1ccccc1Nc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.50
TDP1 Q9NUW8 6/20 0.50
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
KDM4E B2RXH2 5/20 0.50
GAA P10253 3/20 0.50
GLA P06280 2/20 0.50
RECQL P46063 1/20 0.50
ALDH1A1 P00352 10/20 0.48
LMNA P02545 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP2D6 P10635 1/20 0.48
HSD17B10 Q99714 4/20 0.46
ALOX15 P16050 5/20 0.45
HPGD P15428 4/20 0.45
TSHR P16473 3/20 0.45
CYP3A4 P08684 3/20 0.45
TP53 P04637 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31091224 0.86 ALDH1A1 (0.48) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL28410286 0.84 MAPT (0.48) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL31153233 0.84 MAPT (0.48) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL24292255 0.84 MAPK13 (0.40) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL16860103 0.81 MAPT (0.46) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL25502791 0.81 KDM4E (0.42) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL14349843 0.80 MAPT (0.44) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL292427 0.80 MAPT (0.44) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL291442 0.80 MAPT (0.44) MAPTTDP1MEN1KMT2AKDM4E
SCHEMBL27651007 0.80 MAPT (0.53) MAPTTDP1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 134 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6111045-A YIELDS A VULCANIZED RUBBER SHOWING IMPROVEMENTS IN HEAT BUILD-UP, TENSILE STRENGTH, ABRASION RESISTANCE AND PROCESSABILITY NIPPON ZEON CO. LTD. (JP) 2000-08-29 US claimed
JP-61130355-A None JP disclosed
CN-114671825-A Synthetic method of chiral 4H-3, 1-benzoxazine compound containing selenium aryl 安徽泽升科技有限公司 2022-06-28 CN disclosed
EP-3851489-A1 MODIFIED MULTI-COMPONENT COPOLYMER, RUBBER COMPOSITION, RESIN COMPOSITION, TIRE AND RESIN PRODUCT BRIDGESTONE CORPORATION (JP) 2021-07-21 EP disclosed
WO-2020054484-A1 MODIFIED MULTI-COMPONENT COPOLYMER, RUBBER COMPOSITION, RESIN COMPOSITION, TIRE AND RESIN PRODUCT 株式会社ブリヂストン 2020-03-19 WO disclosed
US-20180244808-A1 METHOD FOR PRODUCING MODIFIED DIENE-BASED RUBBER, RUBBER COMPOSITION AND TIRE BRIDGESTONE CORPORATION (JP) 2018-08-30 US disclosed
EP-3345933-A1 METHOD FOR PRODUCING MODIFIED DIENE RUBBER, RUBBER COMPOSITION, AND TIRE Bridgestone Corporation (JP) 2018-07-11 EP disclosed
EP-3029099-B1 RUBBER COMPOSITION AND TIRE PRODUCED USING SAME, AND PROCESS OF PRODUCING RUBBER COMPOSITION BRIDGESTONE CORP (JP) 2018-04-04 EP disclosed
EP-2845869-B1 MODIFIED NATURAL RUBBER, METHOD FOR PRODUCING SAME, RUBBER COMPOSITION, AND TIRE BRIDGESTONE CORP (JP) 2018-01-17 EP disclosed
EP-2799482-B1 Rubber composition and tire produced using same, and process of producing rubber composition BRIDGESTONE CORP (JP) 2017-03-29 EP disclosed
US-6114432-A A DIENE RUBBER COMPONENT INCLUDING AN AMINO GROUP-CONTAINING VINYL MONOMER REINFORCED WITH SILICA; AUTOMOBILE TIRES HAVING EXCELLENT HEAT BUILD-UP RESISTANCE, TENSILE PROPERTIES, ABRASION PROPERTIES AND PROCESSIBILITY NIPPON ZEON CO., LTD. (JP) 2000-09-05 US disclosed
US-6111045-A YIELDS A VULCANIZED RUBBER SHOWING IMPROVEMENTS IN HEAT BUILD-UP, TENSILE STRENGTH, ABRASION RESISTANCE AND PROCESSABILITY NIPPON ZEON CO. LTD. (JP) 2000-08-29 US disclosed
US-6075092-A DIENE RUBBER AND A SPECIFIED ETHYLENE OXIDE-PROPYLENE OXIDE-UNSATURATED OXIDE TERPOLYMER HAVING GIVEN MOONEY VISCOSITY; EXCELLENT HEAT BUILD-UP RESISTANCE, TENSILE STRENGTH AND PROCESSABILITY NIPPON ZEON CO., LTD. (JP) 2000-06-13 US disclosed
US-6013737-A HAVING IMPROVED TENSILE MODULUS AND IMPROVED ABRASION RESISTANCE, COMPRISING AN AMINO GROUP-CONTAINING DIENE RUBBER OF GIVEN MOONEY VISCOSITY, AND SILICA HAVING SPECIFIC SURFACE AREA, A VULCANIZER AND VULCANIZATION ACCELERATOR NIPPON ZEON CO., LTD. (JP) 2000-01-11 US disclosed
EP-0894824-A1 RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1999-02-03 EP disclosed
EP-0870786-A1 DIENE RUBBER, PROCESS FOR THE PREPARATION OF THE SAME AND COMPOSITION CONTAINING THE SAME NIPPON ZEON CO., LTD. (JP) 1998-10-14 EP disclosed
EP-0864606-A1 RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1998-09-16 EP disclosed
EP-0849321-A1 DIENE RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1998-06-24 EP disclosed
EP-0819731-A1 DIENE RUBBER COMPOSITION NIPPON ZEON CO., LTD. (JP) 1998-01-21 EP disclosed
JP-S61130355-A ANTIOXIDANT FOR RUBBER-LIKE POLYMER NIPPON ZEON CO LTD 1986-06-18 JP disclosed