SCHEMBL29200006

SCHEMBL29200006

CCCNC(=O)c1ccc(CNC(=O)c2cc(C(C)C)c(O)cc2O)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 13/20 0.70
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP3A5 P20815 1/20 0.70
CYP3A7 P24462 1/20 0.70
CYP2C19 P33261 1/20 0.70
CYP3A43 Q9HB55 1/20 0.70
HDAC3 O15379 5/20 0.51
HDAC1 Q13547 4/20 0.51
HDAC6 Q9UBN7 3/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HSP90AB1 P08238 1/20 0.48
HDAC2 Q92769 3/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HDAC8 Q9BY41 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25100417 0.87 HDAC6 (0.66) HSP90AA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL20677834 0.82 HSP90AA1 (1.00) HSP90AA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL21644656 0.82 SMN1; SMN2 (0.53) HSP90AA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL21644655 0.81 HSP90AA1 (0.64) HSP90AA1CYP3A4CYP2C9CYP2C19HSP90AB1
SCHEMBL28260522 0.74 HDAC3 (0.78) HDAC3HDAC1HDAC6HDAC7HDAC2
SCHEMBL21644589 0.74 HSP90AA1 (0.48) HSP90AA1HDAC3HDAC1HDAC6HDAC7
SCHEMBL30779607 0.74 HSP90AA1 (0.48) HSP90AA1HDAC3HDAC1HDAC6HDAC7
SCHEMBL19183432 0.73 HSP90AA1 (1.00) HSP90AA1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28867177 0.73 MAPK1 (0.60) HDAC3HDAC1HDAC6HDAC7HDAC2
SCHEMBL14368640 0.71 HSP90AA1 (0.46) HSP90AA1CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112661661-B Compounds having HSP90 inhibitory activity or pharmaceutically acceptable salts thereof and medical use thereof 恩科森株式会社 2023-06-27 CN disclosed