SCHEMBL28260522

SCHEMBL28260522

CCCNC(=O)c1ccc(CNC(=O)c2ccccc2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 9/20 0.78
HDAC1 Q13547 8/20 0.78
HDAC2 Q92769 6/20 0.78
HDAC6 Q9UBN7 5/20 0.69
HDAC8 Q9BY41 2/20 0.61
LMNA P02545 2/20 0.60
RAB9A P51151 1/20 0.60
EPHX2 P34913 1/20 0.60
NR1H4 Q96RI1 1/20 0.60
POLB P06746 2/20 0.60
KDM4E B2RXH2 1/20 0.60
TSHR P16473 1/20 0.60
RECQL P46063 1/20 0.60
PPARG P37231 1/20 0.59
NAAA Q02083 1/20 0.59
HDAC4 P56524 1/20 0.59
HDAC7 Q8WUI4 1/20 0.59
HDAC10 Q969S8 1/20 0.59
HDAC11 Q96DB2 1/20 0.59
HDAC9 Q9UKV0 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21435753 0.88 HDAC3 (1.00) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL334957 0.88 NAAA (0.73) HDAC3HDAC1HDAC2HDAC6HDAC8
Benzene SCHEMBL28248159 0.88 NAAA (0.73) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL11341368 0.86 NAAA (0.71) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL11338329 0.86 NAAA (0.71) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL11348229 0.86 NAAA (0.71) HDAC3HDAC1HDAC2HDAC6HDAC8
Hydrochloric Acid SCHEMBL7763902 0.86 NAAA (0.71) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL28867177 0.86 MAPK1 (0.60) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL1927473 0.85 RAB9A (0.67) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL1926268 0.85 HDAC2 (0.58) HDAC3HDAC1HDAC2HDAC6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884021-A Novel compound having HSP90 inhibitory activity or pharmaceutically acceptable salt thereof and medical use thereof 启明大学校产学协力团 2018-11-23 CN disclosed