SCHEMBL29200075

SCHEMBL29200075

CONC(=O)[C@@H]1CC(c2ccc(C(F)(F)F)cc2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 1/20 0.51
POLB P06746 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
F2R P25116 3/20 0.41
MAPT P10636 1/20 0.40
TACR1 P25103 8/20 0.40
RORC P51449 1/20 0.40
CETP P11597 1/20 0.39
HSD11B1 P28845 1/20 0.39
P2RY14 Q15391 1/20 0.39
STS P08842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184744 0.88 HTRA1 (0.46) HTRA1POLBKDM4EALDH1A1GAA
SCHEMBL28529255 0.85 HTRA1 (0.48) HTRA1F2RMAPTTACR1RORC
SCHEMBL24645690 0.85 HTRA1 (0.48) HTRA1F2RMAPTTACR1RORC
SCHEMBL6183705 0.85 HTRA1 (0.48) HTRA1F2RMAPTTACR1RORC
SCHEMBL28531769 0.82 TACR1 (0.42) HTRA1POLBF2RMAPTTACR1
SCHEMBL28537494 0.81 TACR1 (0.46) HTRA1F2RMAPTTACR1RORC
SCHEMBL28531832 0.80 CYP3A4 (0.42) POLBKDM4EALDH1A1GAAMAPK1
SCHEMBL28536977 0.78 TACR1 (0.43) HTRA1POLBKDM4EALDH1A1GAA
SCHEMBL28539977 0.78 TACR1 (0.43) HTRA1POLBKDM4EALDH1A1GAA
SCHEMBL21619693 0.77 TACR1 (0.48) MAPTTACR1RORCCETPP2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed