SCHEMBL28537494

SCHEMBL28537494

CCN(C)C(=O)[C@@H]1CC(c2ccc(C(F)(F)F)cc2)CN1C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.46
HTRA1 Q92743 1/20 0.43
CETP P11597 2/20 0.42
MAPT P10636 1/20 0.39
GHSR Q92847 1/20 0.39
RORC P51449 4/20 0.39
F2R P25116 2/20 0.38
P2RY14 Q15391 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28531769 0.86 TACR1 (0.42) TACR1HTRA1CETPMAPTRORC
SCHEMBL6184744 0.84 HTRA1 (0.46) TACR1HTRA1CETPMAPTRORC
SCHEMBL28529255 0.83 HTRA1 (0.48) TACR1HTRA1MAPTRORCF2R
SCHEMBL24645690 0.83 HTRA1 (0.48) TACR1HTRA1MAPTRORCF2R
SCHEMBL6183705 0.83 HTRA1 (0.48) TACR1HTRA1MAPTRORCF2R
SCHEMBL29200075 0.81 HTRA1 (0.51) TACR1HTRA1CETPMAPTRORC
SCHEMBL28532292 0.80 CETP (0.48) TACR1CETPMAPTRORCP2RY14
SCHEMBL28532289 0.80 CETP (0.48) TACR1CETPMAPTRORCP2RY14
SCHEMBL21619693 0.78 TACR1 (0.48) TACR1CETPMAPTRORCP2RY14
SCHEMBL28537130 0.78 TACR1 (0.44) TACR1CETPMAPTRORCF2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed