SCHEMBL29200857

SCHEMBL29200857

NC(=O)C1CC(C(N)=O)N(c2ccncn2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 1/20 0.37
CTSS P25774 1/20 0.37
CHRM1 P11229 1/20 0.35
GPR119 Q8TDV5 1/20 0.34
PARP1 P09874 2/20 0.34
RIPK1 Q13546 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
CYP2D6 P10635 1/20 0.34
DPP4 P27487 1/20 0.34
KCNH2 Q12809 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
CHRM4 P08173 2/20 0.33
LSS P48449 1/20 0.33
AKT1 P31749 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
SORD Q00796 1/20 0.33
P2RX7 Q99572 1/20 0.33
RPS6KA5 O75582 1/20 0.32
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30475254 1.00 GRM1 (0.37) GRM1CTSSCHRM1GPR119PARP1
SCHEMBL29200964 0.82 GRM1 (0.41) GRM1CTSSCYP2D6
SCHEMBL29851199 0.78 GPBAR1 (0.44) GRM1CHRM1GPR119PARP1RIPK1
SCHEMBL1381113 0.74 GPR119 (0.36) GRM1CHRM1GPR119PARP1RIPK1
SCHEMBL29200952 0.74 KDM4E (0.60) CNR2
SCHEMBL29200928 0.73 CTSS (0.33) CTSS
SCHEMBL9108658 0.73 GAA (0.45) GRM1CTSSCHRM1GPR119RIPK1
SCHEMBL29200927 0.71 CHRNA4 (0.35) CTSSEPHX2
SCHEMBL1290812 0.71 GPBAR1 (0.57) GRM1GPR119RIPK1GPBAR1CYP2D6
SCHEMBL29200861 0.70 KDM4C (0.44) GRM1DPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332905-A (S) -N-phenyl-1- (pyridin-2-yl) pyrrolidine-2-carboxamide derivatives 上海翊石医药科技有限公司 2023-06-27 CN disclosed