SCHEMBL29208124

SCHEMBL29208124

CCc1c(I)sc2c(Br)cccc12

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PRNP P04156 1/20 0.34
PSMB8 P28062 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30184539 1.00 PRNP (0.34) PRNPPSMB8GABRA1GABRB2ALDH1A1
SCHEMBL31107739 0.79
SCHEMBL30640501 0.70 NPC1 (0.45) ALDH1A1MEN1KMT2A
SCHEMBL8038388 0.70 PSMB8 (0.33) PSMB8GABRA1GABRB2ALDH1A1
SCHEMBL11933059 0.70 PSMB8 (0.43) PRNPPSMB8ALDH1A1
SCHEMBL31107782 0.69 PIM1 (0.32) PSMB8ALDH1A1MEN1KMT2A
SCHEMBL27002569 0.69 DYRK1A (0.37) PSMB8ALDH1A1MEN1KMT2A
SCHEMBL17207338 0.68 AHR (0.36) PSMB8
SCHEMBL10432656 0.68 PSMB8 (0.36) PSMB8GABRA1GABRB2ALDH1A1
SCHEMBL1293277 0.68 GABRA1 (0.48) PRNPGABRA1GABRB2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240400591-A1 COMPOUNDS TARGETING MUTANT OF P53 JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2024-12-05 US disclosed
CN-117986235-A P53-Y220C selective small molecule reactivation agent compound, pharmaceutical composition and application thereof 长春金赛药业有限责任公司 2024-05-07 CN disclosed
CN-117813295-A Compounds targeting p53 mutants 北京加科思新药研发有限公司 2024-04-02 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240400591-A1 COMPOUNDS TARGETING MUTANT OF P53 TP53, TP53BP1, MDM2 PRNP 1337/4885PSMB8 1717/4885GABRA1 4552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.