SCHEMBL292108

SCHEMBL292108

Clc1nc2c(N3CCC3)nc(N3CCNCC3)nc2nc1OOCCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 15/20 0.60
PDE4B Q07343 15/20 0.60
PDE4C Q08493 15/20 0.60
PDE4D Q08499 15/20 0.60
CETP P11597 3/20 0.41
HTR2C P28335 1/20 0.38
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292370 0.91 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL357498 0.77 PDE4A (0.48) PDE4APDE4BPDE4CPDE4D
SCHEMBL291798 0.77 PDE4A (0.96) PDE4APDE4BPDE4CPDE4D
SCHEMBL3322406 0.75 PDE4A (0.78) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL292710 0.75 PDE4A (1.00) PDE4APDE4BPDE4CPDE4D
SCHEMBL29824397 0.75 PDE4A (1.00) PDE4APDE4BPDE4CPDE4D
SCHEMBL3322237 0.71 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DHTR2C
SCHEMBL3322428 0.71 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DHTR2C
SCHEMBL6397973 0.71 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DHTR2C
SCHEMBL10709061 0.70 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029600-B1 SUBSTITUTED PTERIDINES SUBSTITUTED WITH A FOUR-MEMBERED HETEROCYCLE BOEHRINGER INGELHEIM INT (DE) 2012-03-14 EP disclosed