SCHEMBL29213685

SCHEMBL29213685

O=c1[nH]c2ccc([N+](=O)[O-])nc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GALR3 O60755 1/20 0.51
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
PDE3B Q13370 9/20 0.41
PDE3A Q14432 9/20 0.41
PDE2A O00408 2/20 0.41
P2RY12 Q9H244 1/20 0.40
TYRO3 Q06418 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
APEX1 P27695 1/20 0.39
KMT2A Q03164 1/20 0.39
HTT P42858 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.37
BCL6 P41182 1/20 0.37
BCOR Q6W2J9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1586090 0.71 PDE3B (0.47) PDE3BPDE3APDE2AP2RY12TYRO3
SCHEMBL5786187 0.69 SIRT2 (0.60) GALR3KDM4EPDE3BPDE3APDE2A
SCHEMBL1502964 0.69 PDE3B (0.50) KDM4EPDE3BPDE3APDE2AP2RY12
SCHEMBL1592898 0.66 KDM4E (0.41) KDM4EGAAMAPTMEN1KMT2A
SCHEMBL16939766 0.66 PDE3B (0.44) PDE3BPDE3APDE2AP2RY12TYRO3
SCHEMBL1163700 0.66 SIRT2 (0.64) PDE3BPDE3APDE2AP2RY12TYRO3
SCHEMBL29703027 0.64 PDE3B (0.41) PDE3BPDE3APDE2AP2RY12TYRO3
SCHEMBL8014109 0.64 KDM4E (0.43) KDM4EGAAMAPTMEN1APEX1
SCHEMBL20777269 0.64 ADORA3 (0.57) KDM4EGAAPDE3BPDE3APDE2A
SCHEMBL1842652 0.64 GRIA1 (0.79) CA12CA9MAPTMEN1APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117820236-A Histone acetyltransferase small molecule inhibitor and preparation method and application thereof 复旦大学 2024-04-05 CN disclosed