SCHEMBL292137

SCHEMBL292137

[CH2]Cc1nc2ccccc2o1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.70
RAB9A P51151 6/20 0.70
MAPT P10636 4/20 0.70
TP53 P04637 5/20 0.63
SMN1; SMN2 Q16637 5/20 0.63
LMNA P02545 1/20 0.63
LOXL2 Q9Y4K0 1/20 0.61
HTT P42858 1/20 0.53
GFER P55789 1/20 0.53
ALOX5 P09917 1/20 0.46
PSMB8 P28062 1/20 0.46
NPSR1 Q6W5P4 2/20 0.44
USP2 O75604 1/20 0.44
DDAH1 O94760 1/20 0.43
ADRA2C P18825 1/20 0.43
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5538025 0.84 MAPT (0.78) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL1420033 0.83 TP53 (0.81) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL155002 0.83 MAPT (1.00) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL5543729 0.81 MAPT (0.72) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL5537492 0.80 MAPT (0.76) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL9642061 0.79 MAPT (0.84) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL2621291 0.79 MAPT (0.70) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL2792617 0.79 NPC1 (0.70) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL622536 0.79 NPC1 (0.70) NPC1RAB9AMAPTTP53SMN1; SMN2
SCHEMBL1786789 0.79 LOXL2 (0.72) NPC1RAB9AMAPTTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 168 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107759532-A A kind of the ethyl 9 oxime derivate of benzoxazole 2, its preparation method and application 苏州大学 2018-03-06 CN claimed
EP-2091929-A1 AGENTS THAT DISRUPT CELLULAR REPLICATION AND THEIR USE IN INHIBITING PATHOLOGICAL CONDITIONS The European Molecular Biology Laboratory (DE) 2009-08-26 EP claimed
CN-101421257-A Agents that disrupt cellular replication and their use in inhibiting pathological conditions EUROPEAN MOLECULAR BIOLOGY LAB EMBL (DE) 2009-04-29 CN claimed
WO-2007107352-A1 AGENTS THAT DISRUPT CELLULAR REPLICATION AND THEIR USE IN INHIBITING PATHOLOGICAL CONDITIONS THE EUROPEAN MOLECULAR BIOLOGY LABORATORY (DE) 2007-09-27 WO claimed
CN-111511465-B Method for producing organic silicon dioxide material and use thereof 埃克森美孚科技工程公司 2023-06-06 CN disclosed
US-11661410-B2 Tricyclic compounds as histone methyltransferase inhibitors GLOBAL BLOOD THERAPEUTICS, INC. (US) 2023-05-30 US disclosed
US-11584734-B2 Tricyclic compounds as histone methyltransferase inhibitors GLOBAL BLOOD THERAPEUTICS, INC. (US) 2023-02-21 US disclosed
US-20230002351-A1 TRICYCLIC COMPOUNDS AS HISTONE METHYLTRANSFERASE INHIBITORS GLOBAL BLOOD THERAPEUTICS, INC. 2023-01-05 US disclosed
US-11325111-B2 Catalysts and methods of making the same EXXONMOBIL RESEARCH & ENGINEERING COMPANY (US) 2022-05-10 US disclosed
CN-109311001-B Organosilica polymer catalyst and method for producing same 埃克森美孚研究工程公司 2022-04-08 CN disclosed
US-11111352-B2 Methods of producing organosilica materials and uses thereof EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2021-09-07 US disclosed
CN-107001945-B Aromatic hydrogenation catalyst and use thereof 埃克森美孚研究工程公司 2020-12-18 CN disclosed
WO-1996040141-A1 4,5-BRIDGED QUINOXALINEDIONES AND QUINOLONES AND THE USE THEREOF AS EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ACEA PHARMACEUTICALS, INC. (US) 1996-12-19 WO disclosed
EP-0642508-A1 TRICYCLIC QUINOXALINEDIONES AS GLUTAMATE RECEPTOR ANTAGONISTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1995-03-15 EP disclosed
WO-1993008188-A1 TRICYCLIC QUINOXALINEDIONES AS GLUTAMATE RECEPTOR ANTAGONISTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1993-04-29 WO disclosed
US-4576753-A MICROBIOCIDES, ANTIBIOTICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1986-03-18 US disclosed
US-4472309-A ANTIMICROBIAL FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-09-18 US disclosed
US-4304718-A ANTIBIOTICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-12-08 US disclosed
US-4264498-A REACTED WITH AN ACID, ITS ACID HALIDE, OR ANHYDRIDE IN THE PRESENCE OF BORON TRIHALIDE AND AN ORGANIC BASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-04-28 US disclosed
US-4181800-A ANTIBIOTICS FROM SUBSTITUTED PERHYDRO-S-TRIAZINES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-01-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230002351-A1 TRICYCLIC COMPOUNDS AS HISTONE METHYLTRANSFERASE INHIBITORS EHMT1, EHMT2, BMI1 NPC1 2406/4885RAB9A 1696/4885MAPT 2437/4885
US-11661410-B2 Tricyclic compounds as histone methyltransferase inhibitors EHMT1, EHMT2, BMI1 NPC1 2406/4885RAB9A 1696/4885MAPT 2437/4885
US-11325111-B2 Catalysts and methods of making the same CAT, STOM, SOD1 NPC1 1201/4885RAB9A 2386/4885MAPT 2655/4885
US-11584734-B2 Tricyclic compounds as histone methyltransferase inhibitors EHMT1, EHMT2, BMI1 NPC1 2468/4885RAB9A 1619/4885MAPT 2954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.