SCHEMBL29237779

SCHEMBL29237779

O=C1c2cccc(Br)c2CC1(F)I

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.42
PIM1 P11309 1/20 0.42
CSNK1A1 P48729 1/20 0.42
ROCK1 Q13464 1/20 0.42
DYRK1A Q13627 1/20 0.42
LRRK2 Q5S007 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
PARP10 Q53GL7 1/20 0.40
PARP11 Q9NR21 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GSK3B P49841 1/20 0.31
CDK5R1 Q15078 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25003063 0.82 CDK5 (0.44) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL29237769 0.79 NSD2 (0.36) CDK5CCNB2CDK1CCNB1GSK3B
SCHEMBL29237856 0.76 PIM1 (0.39) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL29237858 0.76 PIM1 (0.39) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL22989994 0.75 CDK5 (0.44) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL29237837 0.72 CA1 (0.39) CA1CA2CA7CA9
SCHEMBL29237766 0.71 KDM4E (0.38) CA1CA2CA7CA9
SCHEMBL29237787 0.71 NPSR1 (0.47) CA1CA2CA7CA9
SCHEMBL14938952 0.70 CDK5 (0.40) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL28502513 0.70 PARP10 (0.45) CDK5PIM1CSNK1A1ROCK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118239862-A Chiral monofluorone carbonyl substituted nitrile compound and preparation method and application thereof 上海应用技术大学 2024-06-25 CN disclosed