SCHEMBL14938952

SCHEMBL14938952

O=C1c2cccc(Br)c2CC1(Br)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 2/20 0.40
PIM1 P11309 1/20 0.40
CSNK1A1 P48729 1/20 0.40
ROCK1 Q13464 1/20 0.40
DYRK1A Q13627 1/20 0.40
LRRK2 Q5S007 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
PARP10 Q53GL7 1/20 0.38
PARP11 Q9NR21 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
HSP90AA1 P07900 1/20 0.35
CFTR P13569 1/20 0.34
GOPC Q9HD26 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939135 0.83 ALDH1A1 (0.40) PARP10PARP11CA1CA2CA7
SCHEMBL14939641 0.83 MAPT (0.34) CDK5CFTRGOPCGAAMAPT
SCHEMBL14938950 0.83 SRD5A1 (0.36) CA1CA2CA7CA9CFTR
SCHEMBL14939637 0.79 ACHE (0.43) CA1CA2CA7CA9MAPT
SCHEMBL14938940 0.76 NPSR1 (0.49) CFTRGOPCGAAMAPTRAB9A
SCHEMBL22989994 0.73 CDK5 (0.44) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL25003063 0.73 CDK5 (0.44) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL29237779 0.70 CDK5 (0.42) CDK5PIM1CSNK1A1ROCK1DYRK1A
SCHEMBL14939470 0.70 L3MBTL1 (0.41) LRRK2PARP10PARP11CA1CA2
SCHEMBL14938921 0.70 TDP1 (0.47) CDK5LRRK2PARP10CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed