SCHEMBL29238908

SCHEMBL29238908

COc1cncc(-c2cc(C)nc(C(=O)O)c2)c1C

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.46
KDM4E B2RXH2 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALOX15 P16050 1/20 0.40
ACVR1 Q04771 6/20 0.38
TGFBR1 P36897 5/20 0.38
LMNA P02545 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ECE1 P42892 2/20 0.36
ALDH1A1 P00352 3/20 0.36
CNR2 P34972 1/20 0.35
MCL1 Q07820 1/20 0.34
KMO O15229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29238864 0.81 CYP11B2 (0.45)
SCHEMBL4771510 0.78 ALOX15 (0.51) GPR35KDM4EL3MBTL1ALOX15TDP1
SCHEMBL4772437 0.75 MKNK1 (0.49) KDM4EALDH1A1MCL1
SCHEMBL29238863 0.74 PRKCQ (0.36) KDM4EACVR1TGFBR1
SCHEMBL4769459 0.73 DHODH (0.49)
SCHEMBL4772052 0.72 ALOX15 (0.46) GPR35KDM4EALOX15LMNATDP1
SCHEMBL4778161 0.71 HCAR2 (0.47) GPR35KDM4EALOX15ALDH1A1MCL1
SCHEMBL4779431 0.70 HCAR2 (0.39) GPR35KDM4EALOX15ALDH1A1MCL1
SCHEMBL4769103 0.70 MCL1 (0.64) KDM4EL3MBTL1ALDH1A1MCL1
SCHEMBL4778496 0.70 ABL1 (0.41) GPR35KDM4EALOX15TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118251390-A Heteroaryl linked analogs as MGLU5 negative allosteric modulators and methods of making and using the same 范德比尔特大学 2024-06-25 CN disclosed