SCHEMBL29244608

SCHEMBL29244608

O=C(O)c1ccc(COc2ccnc3[nH]ccc23)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXRA P19793 7/20 0.50
RXRB P28702 6/20 0.47
RXRG P48443 5/20 0.47
HPGD P15428 2/20 0.47
MRGPRX4 Q96LA9 1/20 0.45
RHEB Q15382 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
IKBKB O14920 1/20 0.44
CHUK O15111 1/20 0.44
FOLH1 Q04609 1/20 0.44
NUDT1 P36639 1/20 0.44
POLB P06746 2/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
PPIA P62937 1/20 0.43
NEK1 Q96PY6 1/20 0.43
NR4A2 P43354 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2999856 0.83 AURKB (0.51) IKBKBCHUKNUDT1POLBMAPT
SCHEMBL29244612 0.78 PRKCI (0.42) IKBKBCHUKNUDT1
SCHEMBL31072687 0.76 RXRA (0.56) RXRARXRBRXRGHPGDMRGPRX4
SCHEMBL2310574 0.74 NUDT1 (0.49) IKBKBCHUKNUDT1
SCHEMBL29244676 0.74 JAK1 (0.41) HPGDSMN1; SMN2IKBKBCHUKMAPT
SCHEMBL4791827 0.73 IKBKB (0.76) IKBKBCHUKNUDT1NEK1
SCHEMBL4365456 0.71 AURKB (0.56) IKBKBCHUK
SCHEMBL2992617 0.70 NUDT1 (0.55) HPGDSMN1; SMN2IKBKBCHUKNUDT1
SCHEMBL367358 0.70 MRGPRX4 (0.54) RXRARXRBRXRGHPGDMRGPRX4
SCHEMBL27616079 0.70 NUDT1 (0.51) IKBKBCHUKNUDT1NEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118239926-A TLR7 and 8 inhibitors, preparation method and application thereof 上海深势唯思科技有限责任公司 2024-06-25 CN disclosed