SCHEMBL29244643

SCHEMBL29244643

COC(=O)c1ccc(CN)c(=O)n1C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.41
NPC1 O15118 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.39
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.36
BRD4 O60885 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA3 P34903 1/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29244669 0.84 NPC1 (0.40) NPC1NPSR1KDM4EMAPK1ATM
SCHEMBL2176691 0.78 LOXL2 (0.44) LOXL2NPC1NPSR1KDM4EMAPK1
SCHEMBL29244609 0.77 KAT2B (0.36) NPC1NPSR1KDM4EMAPK1ATM
SCHEMBL69407 0.76 KDM4E (0.53) NPC1NPSR1KDM4EMAPK1ATM
SCHEMBL29244595 0.76 NPC1 (0.48) NPC1NPSR1KDM4EMAPK1ATM
SCHEMBL31172759 0.75 HDAC1 (0.41) NPC1NPSR1KDM4EBRD4MAPT
SCHEMBL16653480 0.75 NPC1 (0.47) NPC1NPSR1KDM4EMAPK1ATM
SCHEMBL30935952 0.74 LOXL2 (0.41) LOXL2NPC1KDM4EL3MBTL1ALDH1A1
SCHEMBL8108945 0.72 NPC1 (0.46) NPC1NPSR1KDM4EMAPK1ATM
SCHEMBL7860405 0.70 NPC1 (0.47) NPC1NPSR1KDM4EMAPK1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118239926-A TLR7 and 8 inhibitors, preparation method and application thereof 上海深势唯思科技有限责任公司 2024-06-25 CN disclosed