SCHEMBL29245339

SCHEMBL29245339

C[C@H]1C(Oc2ccc(C(=O)NC3CC3)nc2)CN1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRKAA2 P54646 10/20 0.42
GPR119 Q8TDV5 1/20 0.41
PRKAB2 O43741 5/20 0.41
PRKAG1 P54619 5/20 0.41
PRKAA1 Q13131 5/20 0.41
PRKAG3 Q9UGI9 5/20 0.41
PRKAG2 Q9UGJ0 5/20 0.41
PRKAB1 Q9Y478 5/20 0.41
RAF1 P04049 1/20 0.40
BRAF P15056 1/20 0.40
EPHX2 P34913 1/20 0.40
USP30 Q70CQ3 1/20 0.39
NR3C1 P04150 1/20 0.39
CYP3A4 P08684 1/20 0.39
NAAA Q02083 2/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29245338 1.00 PRKAA2 (0.42) PRKAA2GPR119PRKAB2PRKAG1PRKAA1
SCHEMBL25190399 0.87 HRH3 (0.45) RAF1BRAFEPHX2USP30
SCHEMBL31362178 0.86 USP30 (0.48) PRKAA2GPR119RAF1BRAFEPHX2
SCHEMBL25245422 0.86 USP30 (0.48) PRKAA2GPR119RAF1BRAFEPHX2
SCHEMBL25282936 0.82 GPR119 (0.42) PRKAA2GPR119PRKAB2PRKAG1PRKAA1
SCHEMBL29245342 0.79 USP30 (0.37) GPR119USP30
SCHEMBL29245343 0.79 USP30 (0.37) GPR119USP30
SCHEMBL25607156 0.79 PRKAA2 (0.46) PRKAA2GPR119PRKAB2PRKAG1PRKAA1
SCHEMBL25288882 0.78 PRKAA2 (0.41) PRKAA2GPR119PRKAB2PRKAG1PRKAA1
SCHEMBL25200137 0.77 PRKAA2 (0.57) PRKAA2GPR119PRKAB2PRKAG1PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118019532-A Azetidine and pyrrolidine PARP1 inhibitors and uses thereof 新特拉有限公司 2024-05-10 CN disclosed