SCHEMBL29245342

SCHEMBL29245342

CC1C(Oc2cnc(C(=O)NC3CC3)c(F)c2)CN1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 3/20 0.37
PARP1 P09874 2/20 0.37
HPGDS O60760 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
RIPK2 O43353 3/20 0.35
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4D Q08499 2/20 0.35
RIPK1 Q13546 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
GPR119 Q8TDV5 3/20 0.33
GABRA1 P14867 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
KCNH2 Q12809 1/20 0.33
HPGD P15428 1/20 0.33
PDE4C Q08493 1/20 0.33
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29245343 1.00 USP30 (0.37) USP30PARP1HPGDSHRH3RIPK2
SCHEMBL25240426 0.87 USP30 (0.38) USP30PARP1HPGDSRIPK2GPR119
SCHEMBL31362193 0.87 USP30 (0.38) USP30PARP1HPGDSRIPK2GPR119
SCHEMBL29245339 0.79 PRKAA2 (0.42) USP30GPR119
SCHEMBL25604880 0.79 PARP1 (0.38) USP30PARP1HPGDSHRH3RIPK2
SCHEMBL29245338 0.79 PRKAA2 (0.42) USP30GPR119
Hydrochloric Acid SCHEMBL25240102 0.78 PARP1 (0.38) USP30PARP1HPGDSHRH3RIPK2
SCHEMBL25288422 0.76 HPGDS (0.35) USP30PARP1HPGDSHRH3RIPK2
SCHEMBL25192651 0.73 GPR119 (0.35) USP30GPR119
SCHEMBL30234728 0.73 GPR119 (0.35) USP30GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118019532-A Azetidine and pyrrolidine PARP1 inhibitors and uses thereof 新特拉有限公司 2024-05-10 CN disclosed