SCHEMBL29247486

SCHEMBL29247486

CC(C)(C)OC(=O)N1CCN(c2ncnc3[nH]cc(-c4ccccn4)c23)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 5/20 0.55
BTK Q06187 2/20 0.49
LRRK2 Q5S007 7/20 0.48
ROCK2 O75116 3/20 0.47
ROCK1 Q13464 3/20 0.47
CDC42BPB Q9Y5S2 2/20 0.47
AKT1 P31749 1/20 0.47
AKT1S1 Q96B36 1/20 0.47
SMARCA2 P51531 1/20 0.46
SMARCA4 P51532 1/20 0.46
PBRM1 Q86U86 1/20 0.46
GPR119 Q8TDV5 1/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
STK3 Q13188 3/20 0.44
CDC7 O00311 2/20 0.44
MARK3 P27448 2/20 0.44
PLK4 O00444 1/20 0.44
CHEK1 O14757 1/20 0.44
AURKA O14965 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30372597 1.00 KIT (0.55) KITBTKLRRK2ROCK2ROCK1
SCHEMBL29247560 0.87 KIT (0.45) KITBTKROCK2ROCK1CDC42BPB
SCHEMBL29247293 0.86 LIMK2 (0.53) LRRK2ROCK2ROCK1CDC42BPBLIMK1
SCHEMBL29247726 0.86 BTK (0.51) KITBTKROCK2ROCK1CDC42BPB
SCHEMBL30372519 0.86 LIMK2 (0.53) LRRK2ROCK2ROCK1CDC42BPBLIMK1
SCHEMBL30295210 0.86 BTK (0.51) KITBTKROCK2ROCK1CDC42BPB
SCHEMBL29247286 0.86 LIMK2 (0.53) LRRK2ROCK2ROCK1CDC42BPBLIMK1
SCHEMBL29247122 0.86 BTK (0.51) KITBTKROCK2ROCK1CDC42BPB
SCHEMBL16637074 0.85 LRRK2 (0.61) KITBTKLRRK2AKT1AKT1S1
SCHEMBL30295133 0.85 LRRK2 (0.61) KITBTKLRRK2AKT1AKT1S1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118317963-A TRPML modulators, compositions thereof, and methods of use 卡拉韦治疗公司 2024-07-09 CN disclosed