SCHEMBL29248409

SCHEMBL29248409

COC(=O)C(C(C)C)n1cc(-c2ccc(CO)cc2)cn1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 1/20 0.38
CCNC P24863 4/20 0.36
CDK8 P49336 4/20 0.36
CD274 Q9NZQ7 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
NAMPT P43490 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
HDAC2 Q92769 1/20 0.35
ROCK1 Q13464 1/20 0.35
MYLK4 Q86YV6 1/20 0.35
FYN P06241 1/20 0.35
ACHE P22303 2/20 0.34
MGLL Q99685 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25421046 0.89 CD274 (0.38) ADAMTS4CCNCCDK8CD274GRIN1
SCHEMBL21612897 0.75 HTT (0.40) CD274CYP1A2CYP2C9
SCHEMBL25027328 0.74 KDM4E (0.39) ACHE
SCHEMBL25027331 0.73 KDM4E (0.36) ACHE
SCHEMBL25348004 0.69 GPR119 (0.37) CCNCCDK8CD274MKNK1MKNK2
SCHEMBL30519933 0.69 GPR119 (0.37) CCNCCDK8CD274MKNK1MKNK2
SCHEMBL25754081 0.69 EP300 (0.48) CCNCCDK8NAMPTMKNK1MKNK2
SCHEMBL31413896 0.69 JAK2 (0.33) CYP2C9
SCHEMBL26071338 0.68 ACVR2A (0.41)
SCHEMBL12516034 0.67 EPHB4 (0.50) CCNCCDK8NAMPTMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118317774-A Pharmaceutical compositions comprising quinazoline compounds 安斯泰来制药株式会社 2024-07-09 CN disclosed