SCHEMBL29258115

SCHEMBL29258115

O=C(/C=C/c1ccncc1)Nc1ccc(C(=O)NCc2ccccc2OC(F)(F)F)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.52
EPHX2 P34913 5/20 0.51
ROCK2 O75116 2/20 0.51
PPARG P37231 2/20 0.48
HSD17B13 Q7Z5P4 1/20 0.47
MAOB P27338 1/20 0.45
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ROCK1 Q13464 1/20 0.45
CYP2C9 P11712 2/20 0.44
CYP2J2 P51589 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29258119 1.00 NAMPT (0.52) NAMPTEPHX2ROCK2PPARGHSD17B13
SCHEMBL29258633 0.85 EPHX2 (0.59) NAMPTEPHX2ROCK2PPARGMAOB
SCHEMBL29258630 0.85 EPHX2 (0.59) NAMPTEPHX2ROCK2PPARGMAOB
SCHEMBL29258764 0.83 NAMPT (0.59) NAMPTHDAC1
SCHEMBL29258128 0.83 NAMPT (0.64) NAMPTEPHX2ROCK2PPARGHDAC3
SCHEMBL29258125 0.83 NAMPT (0.64) NAMPTEPHX2ROCK2PPARGHDAC3
SCHEMBL29258151 0.82 NAMPT (0.77) NAMPT
SCHEMBL29258096 0.81 ROCK2 (0.68) NAMPTROCK2ROCK1CYP2C9
SCHEMBL29258099 0.81 ROCK2 (0.68) NAMPTROCK2ROCK1CYP2C9
SCHEMBL29258164 0.79 NAMPT (0.57) NAMPTEPHX2MAOBHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118108664-A NAMPT agonist and preparation method and application thereof 中国人民解放军海军军医大学 2024-05-31 CN claimed
CN-118108664-A NAMPT agonist and preparation method and application thereof 中国人民解放军海军军医大学 2024-05-31 CN disclosed