SCHEMBL29267442

SCHEMBL29267442

O=Cc1cnc2cc(C(F)(F)F)ccc2c1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
GSK3A P49840 3/20 0.39
GSK3B P49841 3/20 0.39
CLK4 Q9HAZ1 3/20 0.39
DYRK3 O43781 2/20 0.39
DYRK1A Q13627 2/20 0.39
STK17A Q9UEE5 2/20 0.39
PRKD3 O94806 2/20 0.39
MAP4K4 O95819 2/20 0.39
KDR P35968 2/20 0.39
AURKB Q96GD4 2/20 0.39
PRKD2 Q9BZL6 2/20 0.39
PLK4 O00444 1/20 0.39
CHEK2 O96017 1/20 0.39
FGFR1 P11362 1/20 0.39
CDK2 P24941 1/20 0.39
FLT4 P35916 1/20 0.39
CLK2 P49760 1/20 0.39
LIMK1 P53667 1/20 0.39
CSNK1G2 P78368 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29267445 0.80 GRM5 (0.42) KDM4E
SCHEMBL29267456 0.77 CYP2A6 (0.41) PIM3KDM4E
SCHEMBL9591539 0.77 MAOB (0.46) PARP1GSK3AGSK3BCLK4DYRK3
SCHEMBL9360788 0.77 PARP1 (0.49) PARP1GSK3AGSK3BCLK4DYRK3
SCHEMBL29267433 0.77 PARP1 (0.41) PARP1GSK3AGSK3BCLK4DYRK3
SCHEMBL4466003 0.75 SORT1 (0.46) PARP1GSK3AGSK3BCLK4DYRK3
SCHEMBL25229015 0.74 TDP1 (0.50) PARP1
SCHEMBL28783999 0.74 PARP1 (0.39) PARP1GSK3AGSK3BCLK4DYRK3
SCHEMBL21143432 0.73 EGFR (0.44) PARP1GSK3AGSK3BCLK4DYRK3
SCHEMBL29267463 0.73 ALDH1A1 (0.49) KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118324761-A USP inhibitor, preparation method and application thereof 北京华森英诺生物科技有限公司 2024-07-12 CN disclosed