SCHEMBL29267658

SCHEMBL29267658

COc1cc(C2=CCN(C(=O)OC(C)(C)C)C2)ccc1[N+](=O)[O-]

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
QDPR P09417 1/20 0.41
CHEK1 O14757 8/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 1/20 0.40
NAMPT P43490 1/20 0.40
GRM5 P41594 1/20 0.39
GRM1 Q13255 1/20 0.39
SIRT6 Q8N6T7 1/20 0.39
PDK4 Q16654 1/20 0.38
CFTR P13569 1/20 0.38
MMP13 P45452 1/20 0.37
TBK1 Q9UHD2 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31324785 1.00 QDPR (0.41) QDPRCHEK1ALDH1A1LMNAMAPT
SCHEMBL520721 0.90 QDPR (0.52) QDPRALDH1A1LMNAMAPTNAMPT
SCHEMBL30957987 0.90 QDPR (0.52) QDPRALDH1A1LMNAMAPTNAMPT
SCHEMBL519881 0.82 QDPR (0.43) QDPRALDH1A1LMNAMAPTNAMPT
SCHEMBL3316550 0.81 GRM1 (0.51) QDPRALDH1A1LMNAMAPTNAMPT
SCHEMBL21847033 0.81 CCNT1 (0.45) QDPRALDH1A1LMNAMAPTNAMPT
SCHEMBL14617535 0.81 ALDH1A1 (0.57) ALDH1A1LMNAMAPTNAMPTGRM5
SCHEMBL31111716 0.79 MAPT (0.47) ALDH1A1LMNAMAPTNAMPTGRM5
SCHEMBL17197336 0.79 CCNT1 (0.46) CHEK1ALDH1A1LMNAMAPTSIRT6
SCHEMBL15283571 0.79 NAMPT (0.47) QDPRNAMPTGRM5GRM1PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116903591-A Pyrimidine amine NUAK inhibitor and preparation method and application thereof 特科罗生物科技(成都)有限公司 2023-10-20 CN disclosed