SCHEMBL2926933

SCHEMBL2926933

CS(=O)(=O)c1cnc2c(cc(C(=O)O)n2Cc2ccc(F)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 5/20 0.41
CYP1A2 P05177 7/20 0.41
CYP3A4 P08684 7/20 0.41
CYP2C19 P33261 6/20 0.41
USP2 O75604 5/20 0.41
CYP2C9 P11712 5/20 0.41
CCR2 P41597 4/20 0.41
TBXA2R P21731 2/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
ALDH1A1 P00352 4/20 0.39
TSHR P16473 4/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HPGD P15428 2/20 0.39
ALOX15 P16050 1/20 0.39
HIF1A Q16665 1/20 0.38
ABCB11 O95342 1/20 0.38
CYP2D6 P10635 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2931092 0.89 MAPT (0.47) CYP1A2CYP3A4CYP2C19USP2CYP2C9
SCHEMBL2921287 0.87 CYP3A4 (0.40) CYP1A2CYP3A4CYP2C19USP2CYP2C9
SCHEMBL2925799 0.76 CYP3A4 (0.38) CYP1A2CYP3A4CYP2C19USP2CYP2C9
SCHEMBL2921880 0.76 CYP1A2 (0.38) CYP1A2CYP3A4CYP2C19USP2CYP2C9
SCHEMBL2993976 0.75 CCR2 (0.48) CCR9CCR2ABCB11
SCHEMBL2924383 0.70 CCR2 (0.76) CCR2TBXA2RABCB11
SCHEMBL2929131 0.70 PTGS2 (0.56) PTGDR2ALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL2926815 0.70 TP53 (0.48) CYP1A2CYP3A4CYP2C19USP2CYP2C9
SCHEMBL3119623 0.69 CCR2 (0.55) CCR9CYP1A2CYP3A4CYP2C19USP2
SCHEMBL297540 0.68 CCR2 (0.46) CCR9CCR2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086950-B1 HETEROCYCLIC INDOLE DERIVATIVES AND MONO- OR DIAZAINDOLE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2010-09-29 EP disclosed