SCHEMBL29269477

SCHEMBL29269477

Cc1cc(OCCC2CCCN(C(=O)OC(C)(C)C)C2)cc(CNC(=O)[C@@H](N)CCc2ccccc2)c1C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.45
BCHE P06276 4/20 0.45
USP30 Q70CQ3 2/20 0.40
ACKR3 P25106 1/20 0.40
KAT7 O95251 1/20 0.40
KAT8 Q9H7Z6 1/20 0.40
CYP2C9 P11712 1/20 0.39
EPHX2 P34913 1/20 0.38
YAP1 P46937 2/20 0.38
GPR119 Q8TDV5 1/20 0.37
FPR3 P25089 1/20 0.37
FPR2 P25090 1/20 0.37
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
KDM1A O60341 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29269478 1.00 HTR6 (0.45) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL30283224 1.00 HTR6 (0.45) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269496 0.92 HTR6 (0.44) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269498 0.92 HTR6 (0.44) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL30283249 0.89 HTR6 (0.44) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269459 0.89 HTR6 (0.44) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269458 0.89 HTR6 (0.44) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269372 0.89 HTR6 (0.46) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269374 0.89 HTR6 (0.46) HTR6BCHEUSP30ACKR3KAT7
SCHEMBL29269379 0.88 HTR6 (0.45) HTR6BCHEUSP30ACKR3YAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118251383-A Macrocyclic compounds as proteasome beta subunit type 5 inhibitors 利德探索中心有限公司 2024-06-25 CN disclosed