SCHEMBL2927307

SCHEMBL2927307

Cc1cncc2c1C(=N)N(Cc1ccccc1)S2(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA12 O43570 7/20 0.43
CA9 Q16790 7/20 0.43
MAPT P10636 5/20 0.40
CA1 P00915 4/20 0.38
HSD11B1 P28845 1/20 0.37
RAB9A P51151 1/20 0.36
TSHR P16473 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925298 0.75 CA12 (0.37) CA12CA9MAPTTSHRKMT2A
SCHEMBL28516402 0.70 CA12 (0.57) CA12CA9CA1HSD11B1RAB9A
SCHEMBL4697449 0.70 CA12 (0.38) CA12CA9MAPTCA1HSD11B1
SCHEMBL12292101 0.65 KDM4E (0.46) CA12CA9CA1KMT2ATDP1
SCHEMBL9821407 0.64 CA12 (0.52) CA12CA9MAPTCA1RAB9A
SCHEMBL12292200 0.63 CA12 (0.39) CA12CA9MAPTCA1HSD11B1
SCHEMBL1172438 0.61 CA12 (1.00) CA12CA9CA1KMT2ATDP1
SCHEMBL30527996 0.61 CA12 (1.00) CA12CA9CA1KMT2ATDP1
SCHEMBL21881930 0.59 AKT2 (0.43) MAPTRAB9AKMT2AALDH1A1
SCHEMBL31658296 0.59 CA12 (0.46) CA12CA9MAPTHSD11B1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940849-B1 ISOTHIAZOLOPYRIDIN-3-YLENAMINES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2010-01-27 EP disclosed
EP-2062476-A1 Insecticide compositions containing 2-cyano(het)-aryl sulfonamide compounds and their isomeric forms with improved activity Bayer CropScience AG (DE) 2009-05-27 EP disclosed
WO-2009056229-A1 INSECTICIDAL COMPOSITIONS OF 2-CYANO(HET)-ARYLSULPHONAMIDE COMPOUNDS AND THEIR ISOMERIC FORMS WITH IMPROVED ACTIVITY BAYER CROPSCIENCE AG (DE) 2009-05-07 WO disclosed
US-20080227636-A1 Isothiazolopyridin-3-Ylenamines for Combating Animal Pests BASF SE (DE) 2008-09-18 US disclosed
US-20080227636-A1 Isothiazolopyridin-3-Ylenamines for Combating Animal Pests BASF SE (DE) 2008-09-18 US disclosed
US-20080227636-A1 Isothiazolopyridin-3-Ylenamines for Combating Animal Pests BASF SE (DE) 2008-09-18 US disclosed
EP-1940849-A1 ISOTHIAZOLOPYRIDIN-3-YLENAMINES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2008-07-09 EP disclosed
WO-2007045588-A1 ISOTHIAZOLOPYRIDIN-3-YLENAMINES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2007-04-26 WO disclosed
WO-2007045588-A1 ISOTHIAZOLOPYRIDIN-3-YLENAMINES FOR COMBATING ANIMAL PESTS BASF SE (DE) 2007-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080227636-A1 Isothiazolopyridin-3-Ylenamines for Combating Animal Pests IPO5, PIR, ACHE CA12 4389/4885CA9 3102/4885MAPT 2775/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.