SCHEMBL29282185

SCHEMBL29282185

CCOC(=O)COc1cc2[nH]ccc2cc1Br

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
GAA P10253 2/20 0.43
NOTUM Q6P988 2/20 0.42
TDP1 Q9NUW8 1/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
P2RY12 Q9H244 1/20 0.41
ALDH1A1 P00352 3/20 0.41
CSNK2A1 P68400 1/20 0.40
CASP3 P42574 1/20 0.40
CASP7 P55210 1/20 0.40
CASP9 P55211 1/20 0.40
USP2 O75604 1/20 0.40
PTPN1 P18031 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
PRNP P04156 1/20 0.39
MAPT P10636 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27998211 0.80 TSHR (0.52) TSHRGAAALDH1A1CASP3CASP7
SCHEMBL27190416 0.79 AXL (0.55) TSHRGAAPDE3BPDE3AP2RY12
SCHEMBL4665845 0.77 PDE3B (0.55) GAAPDE3BPDE3AP2RY12ALDH1A1
SCHEMBL15902172 0.77 PDE3B (0.55) TSHRGAAPDE3BPDE3AP2RY12
SCHEMBL13247758 0.74 TSHR (0.54) TSHRGAATDP1ALDH1A1CASP3
SCHEMBL4611453 0.72 MAOA (0.45) TSHRNOTUMALDH1A1
SCHEMBL14721005 0.72 HPGD (0.56) TSHRGAAPDE3BPDE3AP2RY12
SCHEMBL15252019 0.72 F9 (0.49) TSHRALDH1A1CASP3CASP7CASP9
SCHEMBL4493257 0.71 PTPRC (0.49) TSHRALDH1A1PTPN1CYP1A2
SCHEMBL5529529 0.71 GAA (0.74) GAATDP1ALDH1A1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117999265-A Substituted fused bicyclic macrocyclic compounds and related methods of treatment 阿尔克姆斯有限公司 2024-05-07 CN disclosed