SCHEMBL29285140

SCHEMBL29285140

COc1c(F)cc(C=O)c2[nH]ncc12

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
MCL1 Q07820 1/20 0.35
ERN1 O75460 4/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
BRD4 O60885 2/20 0.33
METAP2 P50579 2/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RAF1 P04049 2/20 0.32
BRAF P15056 2/20 0.32
LCK P06239 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24786481 0.76 BRD4 (0.35) KDM4EALDH1A1HPGDBRD4METAP2
SCHEMBL20577534 0.72 AXL (0.37) KDM4EALDH1A1HPGDBRD4METAP2
SCHEMBL21725762 0.70 BRD4 (0.33) KDM4EALDH1A1HPGDBRD4METAP2
SCHEMBL24613002 0.70 BRD4 (0.33) KDM4EALDH1A1HPGDBRD4METAP2
SCHEMBL1014315 0.69 ERN1 (0.39) LMNAERN1KDM4EMETAP2TDP1
SCHEMBL25241637 0.69 AXL (0.37) KDM4EALDH1A1HPGDBRD4METAP2
SCHEMBL2425808 0.69 LMNA (0.41) LMNAERN1KDM4EALDH1A1HPGD
SCHEMBL21196014 0.68 HTT (0.35) KDM4EALDH1A1HPGDBRD4METAP2
SCHEMBL31166894 0.68 ALDH1A1 (0.42) MCL1ERN1KDM4EALDH1A1TSHR
SCHEMBL4655024 0.68 ALDH1A1 (0.42) MCL1ERN1KDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964643-B Pyrrole [2,3-b ] pyridine derivative and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-07-02 CN disclosed
CN-117964643-A Pyrrole [2,3-b ] pyridine derivative and preparation method and application thereof 苏州朗睿生物医药有限公司 2024-05-03 CN disclosed