SCHEMBL2928646

SCHEMBL2928646

COc1cc(N(C(=O)C(F)(F)F)C2CNC2)ccc1Nc1cncc(-c2cc3cc(F)ccc3[nH]2)n1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.37
TTK P33981 4/20 0.36
FLT3 P36888 2/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33
GRIN2B Q13224 1/20 0.33
SYK P43405 1/20 0.32
F3 P13726 1/20 0.31
PIM3 Q86V86 1/20 0.31
AURKA O14965 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927146 0.84 BRAF (0.37) BRAFTTKFLT3CCNA2CDK2
SCHEMBL2960852 0.83 BRAF (0.37) BRAFTTKFLT3CCNA2CDK2
Trifluoroacetic Acid SCHEMBL2928643 0.80 PTK2 (0.39) TTKCCNA2CDK2ALDH1A1AURKA
SCHEMBL2927992 0.79 ALDH1A1 (0.40) BRAFTTKCCNA2CDK2ALDH1A1
SCHEMBL2928408 0.79 PIM3 (0.46) BRAFTTKFLT3CCNA2CDK2
SCHEMBL14269675 0.78 TTK (0.43) BRAFTTKCCNA2CDK2
SCHEMBL13515312 0.76 KDR (0.46) ALDH1A1AURKA
Trifluoroacetic Acid SCHEMBL2928635 0.75 DYRK1A (0.47) TTK
Trifluoroacetic Acid SCHEMBL2960848 0.75 TMEM97 (0.40) CCNA2CDK2
Hydrochloric Acid SCHEMBL2936353 0.75 MKNK1 (0.49) BRAFTTKCCNA2CDK2PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044051-B1 PYRIDINE AND PYRAZINE DERIVATIVES AS MNK KINASE INHIBITORS BIOVITRUM AB PUBL (SE) 2010-01-27 EP disclosed