SCHEMBL2928699

SCHEMBL2928699

CC(=O)N1CCN(Cc2ccc(-c3cc(OC(N)=O)c(NC(N)=O)s3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 9/20 0.59
HRH3 Q9Y5N1 2/20 0.52
MAP3K7 O43318 1/20 0.50
IKBKE Q14164 1/20 0.45
TBK1 Q9UHD2 1/20 0.45
IKBKB O14920 1/20 0.44
RORC P51449 1/20 0.43
CHRM1 P11229 1/20 0.41
HTR2A P28223 1/20 0.41
MCHR1 Q99705 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
KDR P35968 1/20 0.41
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2933039 0.90 CHEK1 (0.73) CHEK1MAP3K7IKBKETBK1IKBKB
SCHEMBL2930060 0.89 CHEK1 (0.70) CHEK1MAP3K7TBK1IKBKBMEN1
SCHEMBL2933445 0.88 CHEK1 (0.72) CHEK1HRH3MAP3K7IKBKBMEN1
SCHEMBL2934362 0.86 CHEK1 (0.58) CHEK1HRH3MAP3K7TBK1IKBKB
SCHEMBL2932566 0.85 CHEK1 (0.57) CHEK1MAP3K7IKBKBMEN1KMT2A
SCHEMBL1927925 0.85 CHEK1 (0.81) CHEK1HRH3MAP3K7IKBKETBK1
SCHEMBL2933336 0.84 CHEK1 (0.56) CHEK1HRH3MAP3K7IKBKBMEN1
SCHEMBL2932338 0.83 CHEK1 (0.55) CHEK1HRH3MAP3K7IKBKBJAK2
SCHEMBL2931062 0.83 CHEK1 (0.59) CHEK1HRH3MAP3K7TBK1IKBKB
SCHEMBL2931228 0.82 CHEK1 (0.51) CHEK1MAP3K7IKBKBJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421074-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP claimed