SCHEMBL2934362

SCHEMBL2934362

NC(=O)Nc1sc(-c2ccc(CN3CCOCC3)cc2)cc1OC(N)=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.58
MAP3K7 O43318 1/20 0.47
HRH3 Q9Y5N1 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TBK1 Q9UHD2 1/20 0.44
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
IKBKB O14920 1/20 0.43
PARP1 P09874 1/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 1/20 0.42
AOC3 Q16853 1/20 0.42
JAK2 O60674 1/20 0.42
JAK3 P52333 1/20 0.42
KCNH2 Q12809 1/20 0.42
HIF1A Q16665 1/20 0.41
EPAS1 Q99814 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2931062 0.96 CHEK1 (0.59) CHEK1MAP3K7HRH3ALDH1A1TBK1
SCHEMBL2932197 0.91 CHEK1 (0.48) CHEK1ALDH1A1IKBKBPARP1NPC1
SCHEMBL2930060 0.91 CHEK1 (0.70) CHEK1MAP3K7ALDH1A1TBK1IKBKB
SCHEMBL2933445 0.90 CHEK1 (0.72) CHEK1MAP3K7HRH3ALDH1A1IKBKB
SCHEMBL2933039 0.88 CHEK1 (0.73) CHEK1MAP3K7TBK1IKBKBPARP1
SCHEMBL2933735 0.88 CHEK1 (0.44) CHEK1MAP3K7JAK2JAK3KCNH2
SCHEMBL2932566 0.87 CHEK1 (0.57) CHEK1MAP3K7ALDH1A1IKBKBRAB9A
SCHEMBL2925535 0.86 JAK2 (0.43) CHEK1HRH3TBK1JAK2JAK3
SCHEMBL2928699 0.86 CHEK1 (0.59) CHEK1MAP3K7HRH3TBK1IKBKB
SCHEMBL2933336 0.86 CHEK1 (0.56) CHEK1MAP3K7HRH3IKBKBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421074-B1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2010-09-29 EP claimed