SCHEMBL2930106

SCHEMBL2930106

COc1ncnc2sc(NC(=O)ON3CCC(NC(C)=O)(c4cccc(C(F)(F)F)c4)CC3)nc12

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.41
ADORA2B P29275 9/20 0.41
ADORA1 P30542 8/20 0.41
TACR3 P29371 1/20 0.35
CCR2 P41597 1/20 0.35
KCNH2 Q12809 1/20 0.35
DGAT1 O75907 1/20 0.35
TRPV1 Q8NER1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1760896 0.90 ADORA2A (0.52) ADORA2AADORA2BADORA1TACR3
SCHEMBL2932713 0.89 ADORA2A (0.49) ADORA2AADORA2BADORA1CCR2KCNH2
SCHEMBL2931382 0.89 ADORA2A (0.41) ADORA2AADORA2BADORA1TRPV1
SCHEMBL2932934 0.84 ADORA2B (0.40) ADORA2AADORA2BADORA1CCR2KCNH2
SCHEMBL2930871 0.82 ADORA2A (0.49) ADORA2AADORA2BADORA1CCR2TRPV1
SCHEMBL3041508 0.82 PHGDH (0.47) ADORA2A
SCHEMBL1760987 0.81 ADORA2A (0.49) ADORA2AADORA2BADORA1TRPV1
SCHEMBL2927982 0.80 ADORA2B (0.47) ADORA2AADORA2BADORA1KCNH2
SCHEMBL2928074 0.80 ADORA2A (0.51) ADORA2AADORA2BADORA1
SCHEMBL1761019 0.79 ADORA2A (0.52) ADORA2AADORA2BADORA1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed