SCHEMBL29313707

SCHEMBL29313707

CC(=O)N1CCC(n2ccn(-c3cc(C(F)(F)F)cc(C(F)(F)F)c3OC(=O)N(C)c3ccc(F)cc3)c2=O)CC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.39
TACR2 P21452 4/20 0.39
TACR3 P29371 2/20 0.35
POLQ O75417 2/20 0.35
CYP3A4 P08684 3/20 0.34
SIGMAR1 Q99720 1/20 0.34
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313708 0.91 POLQ (0.38) TACR1TACR2POLQCYP3A4CYP2C9
SCHEMBL29313703 0.89 TACR1 (0.39) TACR1TACR2POLQ
SCHEMBL29313711 0.86 TACR1 (0.36) TACR1POLQ
SCHEMBL29313695 0.84 POLQ (0.37) POLQ
SCHEMBL29313712 0.83 POLQ (0.35) TACR1TACR2POLQ
SCHEMBL29313696 0.83 POLQ (0.36) TACR1POLQ
SCHEMBL29313743 0.81 POLQ (0.35) POLQ
SCHEMBL29313746 0.81 POLQ (0.35) POLQ
SCHEMBL29313670 0.81 POLQ (0.35) TACR1TACR2POLQ
SCHEMBL29313609 0.79 POLQ (0.40) POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed