SCHEMBL29313930

SCHEMBL29313930

Cc1nc(N(C)C(=O)Oc2c(C(F)(F)F)cc(C(F)(F)F)nc2-c2nccs2)ccc1F

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.32
S1PR1 P21453 1/20 0.32
ECE1 P42892 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313931 0.90 MEN1 (0.31) ECE1MEN1KMT2A
SCHEMBL29313940 0.84 S1PR1 (0.35) S1PR1GPBAR1
SCHEMBL29313948 0.84 POLQ (0.35) S1PR1ECE1GPBAR1MEN1KMT2A
SCHEMBL29313926 0.83 POLQ (0.34) ECE1GPBAR1
SCHEMBL29313928 0.81 POLQ (0.33)
SCHEMBL29313943 0.75 GPBAR1 (0.34) S1PR1GPBAR1MEN1KMT2A
SCHEMBL29313859 0.72 GAA (0.31) GAA
SCHEMBL29313964 0.68 POLQ (0.33) GAAMEN1KMT2A
SCHEMBL29314053 0.67 IMPDH2 (0.36) GPBAR1
SCHEMBL29313937 0.66 POLQ (0.42) S1PR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed